METHOD AND CATALYST FOR SYNTHESISING AZIRIDINE

Abstract

The present invention relates to methods of synthesising aziridines including isotopically labelled aziridines, said methods comprising contacting an imine or one or more precursors thereof with a diazo compound in the presence of a phosphoramide or a phosphoramide-derived catalyst. The present invention also relates to aziridines, modified aziridines and aziridine-derived compounds preparable by the aforementioned methods, and to phosphoramide or phosphoramide-derived catalysts suitable for use in such methods.


Classe Tecnologica

C - Chemistry and Metallurgy

Patent Office

European Patent Office


Numero Deposito

EP 2861559

Anno Deposito

2013

Anno Concessione

2015


Inventori Pugliesi

  • Pesce Paolo

Tutti gli inventori

  • Bew Sean Patrick
  • Thurston Sean Michael
  • Pesce Paolo

Titolari pugliesi

  • Non ci sono titolari pugliesi

Tutti i titolari

  • University Of East Anglia